2014-317 ACTIVATING HIV LATENCY USING DRUG ENCAPSULATED NANOPARTICLES

Case No. 2014-317

 

SUMMARY

UCLA researchers in the Department of Microbiology, Immunology, and Molecular Genetics have devised a novel method to target the HIV virus in patients using nanoparticles loaded with therapeutic agents.

 

BACKGROUND

Contracting HIV (human immunodeficiency virus) can lead to lifelong complications both physically and mentally. Current HIV therapies are aimed towards controlling the amount of viral replication in patients but fail to completely eliminate the virus. Eradicating the virus from patients is difficult due to a latent population of virus that is established soon after infection. These latent viruses are responsible for the quick recovery of viral loads when a patient is taken off an antiviral regime; therefore, patients must be on medication for life. The ability to totally eliminate these latent viruses will be crucial in reaching a virus-free state in patients.

 

INNOVATION

The disclosed method by Dr. Zerome Zack is the first described method of treating HIV by first targeting/activating the latent virus with a nanoparticle, followed by treatment using antivirals. Drugs are loaded onto nanoparticles that can be engineered for cell-targeting, improving efficiency of drug delivery. This novel therapeutic approach offers the potential to completely eliminate the virus from a patient.

 

APPLICATIONS

Therapy option for HIV patients

Drug-loaded nanoparticles can be used in combination with other HIV treatments

Technology can be extrapolated to treat other viral/bacterial infections

 

ADVANTAGES

Targets latent virus as opposed to only active virus

Method has the potential to completely eradicate virus population in patient

Nanoparticles can be engineered to target specific cells

 

STATE OF DEVELOPMENT

The invention is at the experimental/working prototype stage. It has been demonstrated to be effective in preclinical and in in vitro assays.

 

RELATED MATERIALS

Activation of latent HIV using drug-loaded nanoparticles. Kovochich M, Marsden MD, Zack JA. PLoS One. 2011 Apr 5.

Bioengineered vaults: Self-assembling protein shell-lipophilic core nanoparticles for drug delivery. Buehler DC, Marsden MD, Shen S, Toso DB, Wu X, Lu JA, Zhou ZH, Kickhoefer VA, Wender PA, Zack JA, Rome LH. ACS Nano, July 27 2014

 

PATENT STATUS

Patent Pending

Patent Information: