Multilayered drug delivery implants for localized brain tumor therapy

Background

As treatment strategies evolve for brain tumors, especially post-surgical resection, localized therapy is emerging as a promising alternative to systemic drug delivery. The blood-brain barrier, along with the sensitive anatomy of the brain, makes it difficult to achieve effective therapeutic concentrations using traditional methods without risking widespread toxicity. Targeted delivery systems are essential to improve therapeutic efficacy and minimize side effects.

Existing implantable solutions, such as Gliadel® wafers, present a range of challenges including limited drug effective­ness, uncontrolled release, and serious adverse events like seizures, wound healing issues, and localized swelling. These complications often result from poor pharmacokinetic control and unintended drug diffusion into cerebrospinal regions. Achieving uni­directional, sustained delivery directly at the resection site remains a key unmet need in the field of neuro‑oncology.

Technology overview

This technology introduces a multilayered wafer implant for localized brain drug delivery, designed to overcome the limitations of conventional implants. The implant comprises a hydrophilic polymer-lipid matrix for drug incorpora­tion, encased in a hydrophobic outer layer that controls the direction and rate of drug release. This layered architecture ensures precise, unidirec­tional deliv­ery of therapeutic agents such as chemotherapeutics and steroids directly to the surgical site while minimizing leakage into surrounding cerebrospinal fluid.

The combination of materials enables controlled, prolonged drug release tailored to the pharmacological needs of brain tumor treatment. Unlike tradi­tional polyanhydride-based systems, this design reduces the incidence of adverse side effects by maintaining drug concentration at the target site and limiting systemic exposure. The modular platform is also compatible with a range of drug types, offering broad adaptability for future applications in neuro‑oncology and localized CNS therapies.

Benefits

  • Provides unidirectional, sustained drug release to surgical resection sites
  • Minimizes diffusion into cerebrospinal fluid, reducing adverse side effects
  • Enhances local drug concentration for improved tumor suppression
  • Reduces complications associated with current implants such as seizures and edema
  • Compatible with multiple drug types, including chemotherapeutics and anti-inflammatories

Commercial applications

  • Post-resection brain tumor therapy
  • Localized chemotherapeutic and steroid delivery
  • CNS-targeted drug release platforms
  • Adjunctive therapy in neuro-oncology
  • Implantable controlled-release drug systems

Opportunity

  • Addresses shortcomings of existing brain implant technologies through directional, sustained delivery
  • Offers a modular, biocompatible platform adaptable to a variety of therapeutic agents
  • Available for licensing to partners in neurosurgery, oncology, and advanced drug delivery systems

 

Patent Information:
Title App Type Country Serial No. Patent No. File Date Issued Date Expire Date
IMPLANT COMPOSITIONS FOR THE UNIDIRECTIONAL DELIVERY OF ANTI-CANCER COMPOUNDS TO THE BRAIN Utility (Conversion) United States 15/221,827 9,956,172 7/28/2016 5/1/2018 7/28/2036
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National Europe 16748241.3 3328355 7/28/2016 9/1/2021 7/28/2036
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National Australia 2016298210 2016298210 7/28/2016 3/24/2022 7/28/2036
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National Canada 2,993,823 2,993,823 7/28/2016 1/2/2025 7/28/2036
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National Japan 2018-504129 6938462 7/28/2016 9/3/2021 7/28/2036
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National Germany 16748241.3 602016063103.2 7/28/2016 11/22/2021  
Implant Compositions for the Unidirectional Delivery of Therapeutic Compounds to the Brain National United Kingdom 16748241.3 3328355 7/28/2016 11/24/2021  
IMPLANT COMPOSITIONS FOR THE UNIDIRECTIONAL DELIVERY OF THERAPEUTIC COMPOUNDS TO THE BRAIN Divisional United States 15/928,057 10,434,063 3/21/2018 10/8/2019 7/28/2036
Implant Compositions For The Unidirectional Delivery Of Therapeutic Compounds To The Brain Divisional United States 16/593,187 11,229,599 10/4/2019 1/25/2022 7/28/2036