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Covalent ERK inhibitors for suppressing cancer
BI-78D3, a small molecule, covalently binds to ERK1/2’s D-recruitment site, disrupting ERK signaling crucial for cancer cell growth. This shows promise for treating ERK-dependent cancers, including those resistant to BRAF inhibitors. This disrupts ERK signaling crucial for cell proliferation and survival, particularly in certain cancers like...
Published: 11/8/2024   |   Inventor(s): Kevin Dalby, Ramakrishna Edupuganti, Tamer Kaoud, Chelsea Massaro
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Category(s): Life sciences > Therapeutics > Drug delivery, Life sciences > Therapeutics