Methods of Synthesizing γ-AApeptides and Libraries to Inhibit Aβ Protein Aggregates

Competitive Advantages 

  • Aβ protein aggregate inhibition
  • Protein synthesis time is shortened
  • Multiple ligands can be synthesized
  • Applicable towards multiple diseases

Summary

USF researchers have developed an efficient method of making and screening a γ-AApeptide library. This screening method can identify ligands to a target compound, which is helpful in the identification of new molecular probes and drug candidates. Furthermore, this technology also includes a method of protein synthesis that allows many ligands to be synthesized easily and efficiently. Also developed were methods of inhibiting the toxicity of Aβ aggregates towards N2a neuroblastoma cells, as well as methods and compounds for treating Alzheimer's disease and other neurodegenerative diseases that exhibit Aβ protein aggregates.

 

The Novel Molecule HW-155-1 Effectively Inhibits Aβ40 Protein Aggregation at Different Dosages 

 

Desired Partnerships

  • License
  • Sponsored Research
  • Co-Development
Patent Information:
Title App Type Country Serial No. Patent No. File Date Issued Date Expire Date
Methods of Synthesizing ?-AApeptides, ?-AApeptide Building Blocks, ?-AApeptide Libraries, and ?-AApeptide Inhibitors of ?ß40 Aggregates Utility United States 14/914,960 9,645,155 2/26/2016 5/9/2017 2/26/2036